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BX-912

BX-912

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Product Code: 3081
Availability: In Stock
$209.00
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BX912 is a potent and specific PDK1 inhibitor with IC50 of 12 nM, 9- and 105- fold greater selectivity for PDK1 than PKA and PKC, respectively. In comparison to GSK3β, selectivity for PDK1 is 600-fold.

Chemical Name     N-(3-(4-(2-(1H-imidazol-5-yl)ethylamino)-5-bromopyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide

Inhibitors PI3K/Akt/mTOR PDK-1 BX-912 702674-56-4
Biological Activity:
Biological Activity BX912 is a potent and specific PDK1 inhibitor with IC50 of 12 nM, 9- and 105- fold greater selectivity for PDK1 than PKA and PKC, respectively. In comparison to GSK3β, selectivity for PDK1 is 600-fold.
Technical Data:
M.W. 471.35
Formula: <p>C<sub>20</sub>H<sub>23</sub>BrN<sub>8</sub>O</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 702674-56-4
References:
References Feldman RI, et al. J Biol Chem. 2005, 280(20), 19867-19874.

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