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Nepicastat (SYN-117) HCl

Nepicastat (SYN-117) HCl

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Product Code: 3365
Availability: In Stock
$398.00
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Nepicastat (SYN-117) HCl is a potent and selective inhibitor of both bovine and human dopamine-β-hydroxylase with IC50 of 8.5 nM and 9 nM, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors. Phase 2.

Chemical Name (S)-5-(aminomethyl)-1-(5,7-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)-1H-imidazole-2(3H)-thione hydrochloride

Inhibitors Metabolism Hydroxylase Nepicastat (SYN-117) HCl 170151-24-3
Biological Activity:
Biological Activity Nepicastat (SYN-117) HCl is a potent and selective inhibitor of both bovine and human dopamine-β-hydroxylase with IC50 of 8.5 nM and 9 nM, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors. Phase 2.
Technical Data:
M.W.
Formula: <p>C<sub>14</sub>H<sub>15</sub>F<sub>2</sub>N<sub>3</sub>S.HCl</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 170151-24-3
References:
References Stanley WC, et al. Br J Pharmacol. 1997, 121(8), 1803-1809. Stanley WC, et al. J Cardiovasc Pharmacol. 1998, 31(6), 963-970. Sabbah HN, et al. Circulation. 2000, 102(16), 1990-1995. Schroeder JP, et al. Neuropsychopharmacology. 2010, 35(12), 2440-2449.

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