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GSK J4 HCl

GSK J4 HCl

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Product Code: 3159
Availability: In Stock
$209.00
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GSK J4 HCl is a cell permeable prodrug of GSK J1, which is the first selective inhibitor of the H3K27 histone demethylase JMJD3 and UTX with IC50 of 60 nM and inactive against a panel of demethylases of the JMJ family.

Chemical Name : β-Alanine, N-[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-4-pyrimidinyl]-, ethyl ester, hydrochloride (1:1)

Inhibitors Epigenetics Histone demethylases GSK J4 HCl 1373423-53-0(free base)
Biological Activity:
Biological Activity GSK J4 HCl is a cell permeable prodrug of GSK J1, which is the first selective inhibitor of the H3K27 histone demethylase JMJD3 and UTX with IC50 of 60 nM and inactive against a panel of demethylases of the JMJ family.
Technical Data:
M.W. 453.96
Formula: C<sub>24</sub>H<sub>27</sub>N<sub>5</sub>O<sub>2</sub>.HCl
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 1373423-53-0(free base)
References:
References Kruidenier L, et al. Nature, 2012, 488(7411), 404-408.

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