BI 2536

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Product Code: 3063
Availability: In Stock

$259.00

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BI2536 is a potent Plk1 inhibitor with IC50 of 0.83 nM. It shows 4- and 11-fold greater selectivity against Plk2 and Plk3. Phase 2.

Chemical Name: (R)-4-(8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide

Biological Activity:
Biological Activity	BI2536 is a potent Plk1 inhibitor with IC50 of 0.83 nM. It shows 4- and 11-fold greater selectivity against Plk2 and Plk3. Phase 2.
Technical Data:
M.W.	521.66
Formula:	C<sub>28</sub>H<sub>39</sub>N<sub>7</sub>O<sub>3</sub>
Solubility:	DMSO
Purity:	98%
Storage:	-20℃
CAS No:	755038-02-9
References:
References	Steegmaier M, et al. Curr Biol, 2007, 17(4), 316-322. Nappi TC, et al. Cancer Res, 2009, 69(5), 1916-1923.

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