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Olaparib

Olaparib

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Product Code: 3332
Availability: In Stock
$83.00
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Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1/2 with IC50 of 5 nM/1 nM, 300-times less effective against tankyrase-1. Phase 1/2.

Chemical Name 4-(3-(1-(cyclopropanecarbonyl)piperazine-4-carbonyl)-4-fluorobenzyl)phthalazin-1(2H)-one
Inhibitors Epigenetics PARP Olaparib 763113-22-0
Biological Activity:
Biological Activity Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1/2 with IC50 of 5 nM/1 nM, 300-times less effective against tankyrase-1. Phase 1/2.
Technical Data:
M.W. 434.46
Formula: <p><strong>C<sub>24</sub>H<sub>23</sub>FN<sub>4</sub>O<sub>3</sub></strong></p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 763113-22-0
References:
References Menear KA, et al. J Med Chem, 2008, 51(20), 6581-6591. Evers B, et al, Clin Cancer Res, 2008, 14(12), 3916-3925. Rottenberg S, et al, Proc Natl Acad Sci U S A, 2008, 105(44), 17079-17084. Weston VJ, et al, Blood, 2010, 116(22), 4578-4587.

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