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PF-00562271

PF-00562271

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Product Code: 3360
Availability: In Stock
$587.00
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PF-00562271 is the benzenesulfonate salt of PF-562271, which is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs. Phase 1.

Chemical Name N-methyl-N-(3-((2-(2-oxoindolin-5-ylamino)-5-(trifluoromethyl)pyrimidin-4-ylamino)methyl)pyridin-2-yl)methanesulfonamide benzenesulfonate

Inhibitors Cytoskeletal Signaling FAK PF-00562271 939791-38-5
Biological Activity:
Biological Activity PF-00562271 is the benzenesulfonate salt of PF-562271, which is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs. Phase 1.
Technical Data:
M.W. 665.66
Formula: <p>C<sub>21</sub>H<sub>20</sub>F<sub>3</sub>N<sub>7</sub>O<sub>3</sub>S.C<sub>6</sub>H<sub>6</sub>O<sub>3</sub>S</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 939791-38-5

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