PKC Beta Inhibitor

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Product Code: 9785
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An anilino-monoindolylmaleimide compound that is a potent inhibitor of PKCβ isozymes.

Chemical Name: PKC Beta Inhibitor

Biological Activity:
Biological Activity	PKCβ Inhibitor is an anilino-monoindolylmaleimide compound that acts as a potent and ATP-competitive inhibitor of PKCβ isozymes (IC50 = 5 nM and 21 nM for human PKCβII and βI) and displays greater selectivity over PKCα, PKCγ,PKCε (IC50 = 331 nM, > 1 μM, and 2.8 μM, respectively).
Technical Data:
M.W.	411.46
Formula:	C<sub>24</sub>H<sub>21</sub>N<sub>5</sub>O<sub>2</sub>
Solubility:	Soluble in DMSO (100 mg/ml).
Storage:	Store at 4° C
CAS No:	257879-35-9
References:
References	Tanaka, M., et al. 2004. Bioorg. Med. Chem. Lett. 14, 5171. Pubchem ID: 6419755

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