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Sitaxentan sodium

Sitaxentan sodium

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Product Code: 3251
Availability: In Stock
$335.00
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Sitaxentan sodium is a selective endothelin A receptor (ETA) antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively, exhibits 7000-fold selectivity over ETB. Phase 3.

Chemical Name:
3-Thiophenesulfonamide, N-(4-chloro-3-methyl-5-isoxazolyl)-2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]-, sodium salt (1:1)
 

Inhibitors GPCR & G Protein Endothelin Receptor Sitaxentan sodium 210421-74-2
Biological Activity:
Biological Activity Sitaxentan sodium is a selective endothelin A receptor (ETA) antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively, exhibits 7000-fold selectivity over ETB. Phase 3.
Technical Data:
M.W. 476.89
Formula: C<sub>18</sub>H<sub>14</sub>ClN<sub>2</sub>O6S<sub>2</sub>.Na
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 210421-74-2
References:
References Wu C, et al. J Med Chem. 1997, 40(11), 1690-1697. Tilton RG, et al. Pulm Pharmacol Ther. 2000, 13(2), 87-97. Wanebo JE, et al. Neurosurgery. 1998, 43(6), 1409-1417. Holm P. Scand Cardiovasc J Suppl. 1997, 46, 1-40.

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