Rimonabant

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Product Code: 3281
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Rimonabant is a selective antagonist of CB1 with IC50of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.

Chemical Name 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide

Biological Activity:
Biological Activity	Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
Technical Data:
M.W.	463.79
Formula:	<p>C<sub>22</sub>H<sub>21</sub>Cl<sub>3</sub>N<sub>4</sub>O</p>
Solubility:	DMSO
Purity:	98%
Storage:	-20℃
CAS No:	168273-06-1
References:
References	Chu CM, et al, Org Biomol Chem, 2008, 6(18), 3399-3407 Netherland C, et al, Biochem Biophys Res Commun, 2010, 398(4), 671-676. Rinaldi-Carmona M, et al, FEBS Lett, 1994, 350(2-3), 240-244. Santoro A, et al, Int J Cancer, 2009, 125(5), 996-1003. Schafer A, et al, Br J Pharmacol, 2008, 154(5), 1047-1054. Wise LE, et al, Neuropsychopharmacology, 2007, 32(8), 1805-1812.

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