PFI-1

PFI-1

Product Code: 3356
Availability: In Stock
$180.00
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PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM.

Chemical Name Benzenesulfonamide, 2-methoxy-N-(1,2,3,4-tetrahydro-3-methyl-2-oxo-6-quinazolinyl)-

Biological Activity:
Biological Activity PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM.
Technical Data:
M.W. 347.39
Formula: <p>C<sub>16</sub>H<sub>17</sub>N<sub>3</sub>O<sub>4</sub>S</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 1403764-72-6
References:
References Fish PV, et al. J Med Chem, 2012, 55(22), 9831-9837. Cheng Z, et al. Clin Cancer Res, 2013, 19(7), 1-12. KE Lines, et al. Endocrine Abstracts, 2013.

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