Lapatinib (GW-572016) Ditosylate

Lapatinib (GW-572016) Ditosylate

Product Code: 3403
Availability: In Stock
$180.00
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Lapatinib Ditosylate (GW572016, GW2016) is a potent EGFR and ErbB2 inhibitor with IC50 of 10.8 and 9.2 nM, respectively.

Chemical Name N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine,di4-methylbenzenesulfonate

Biological Activity:
Biological Activity Lapatinib Ditosylate (GW572016, GW2016) is a potent EGFR and ErbB2 inhibitor with IC50 of 10.8 and 9.2 nM, respectively.
Technical Data:
M.W. 925.46
Formula: <p>C<sub>29</sub>H<sub>26</sub>ClFN<sub>4</sub>O<sub>4</sub>S.2C<sub>7</sub>H<sub>8</sub>O<sub>3</sub>S</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 388082-77-7
References:
References Rusnak DW, et al. Mol Cancer Ther, 2001, 1(2), 85-94.

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