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OSI-930

OSI-930

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Product Code: 3337
Availability: In Stock
$587.00
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OSI-930 is a potent inhibitor of Kit, KDR and CSF-1R with IC50 of 80 nM, 9 nM and 15 nM, respectively; also potent to Flt-1, c-Raf and Lck and low activity against PDGFRα/β, Flt-3 and Abl. Phase 1.

Chemical name: 

3-((quinolin-4-ylmethyl)amino)-N-(4-(trifluoromethoxy)phenyl)thiophene-2-carboxamide

Inhibitors Protein Tyrosine Kinase c-Kit OSI-930 728033-96-3
Biological Activity:
Biological Activity OSI-930 is a potent inhibitor of Kit, KDR and CSF-1R with IC50 of 80 nM, 9 nM and 15 nM, respectively; also potent to Flt-1, c-Raf and Lck and low activity against PDGFRα/β, Flt-3 and Abl. Phase 1.
Technical Data:
M.W. 443.44
Formula: <p>C<sub>22</sub>H<sub>16</sub>F<sub>3</sub>N<sub>3</sub>O<sub>2</sub>S</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 728033-96-3
References:
References Garton AJ, et al. Cancer Res. 2006, 66(2):1015-1024. Lin HL, et al. Drug Metab Dispos. 2011, 39(2), 345-350.

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