Ilomastat (GM6001, Galardin)

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Product Code: 3429
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$315.00

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GM6001 (galardin, ilomastat) is a broad spectrum matrix metalloprotease (MMP) inhibitor for MMP-1, MMP-2, MMP-3, MMP-7, MMP-8, MMP-9, MMP-12, MMP-14, and MMP-26 with K_i of 0.4 nM, 0.5 nM, 27 nM, 3.7 nM, 0.1 nM, 0.2 nM, 3.6 nM, 13.4 nM, 0.36 nM, respectively.

Chemical Name Butanediamide, N4-hydroxy-N1-[(1S)-1-(1H-indol-3-ylmethyl)-2-(methylamino)-2-oxoethyl]-2-(2-methylpropyl)-, (2R)-

Biological Activity:
Biological Activity	GM6001 (galardin, ilomastat) is a broad spectrum matrix metalloprotease (MMP) inhibitor for MMP-1, MMP-2, MMP-3, MMP-7, MMP-8, MMP-9, MMP-12, MMP-14, and MMP-26 with Ki of 0.4 nM, 0.5 nM, 27 nM, 3.7 nM, 0.1 nM, 0.2 nM, 3.6 nM, 13.4 nM, 0.36 nM, respectively.
Technical Data:
M.W.	388.46
Formula:	<p>C<sub>20</sub>H<sub>28</sub>N<sub>4</sub>O<sub>4</sub></p>
Solubility:	DMSO
Purity:	98%
Storage:	-20℃
CAS No:	142880-36-2
References:
References	Grobelny D, et al. Biochemistry, 1992, 31(31), 7152-714. Leppert D, et al. J Immunol,1995, 154(9), 4379-4389. Schultz GS, et al. Invest Ophthalmol Vis Sci, 1992, 33(12) 3325-3331. Li C, et al. J Am Coll Cardiol, 2002, 39(11), 1852-1858.

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Ilomastat (GM6001, Galardin)

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