RVX-208

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Product Code: 3269
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$117.00

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RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2, about 170-fold selectivity over BD1. Phase 2.

Chemical Name:
4(3H)-Quinazolinone, 2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-

Biological Activity:
Biological Activity	RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2, about 170-fold selectivity over BD1. Phase 2.
Technical Data:
M.W.	370.4
Formula:	C<sub>20</sub>H<sub>22</sub>N<sub>2</sub>O<sub>5</sub>
Solubility:	DMSO
Purity:	98%
Storage:	-20℃
CAS No:	1044870-39-4
References:
References	Picaud S, et al. Proc Natl Acad Sci U S A. 2013, 110(49), 19754-19759. McNeill E. Curr Opin Investig Drugs. 2010, 11(3), 357-364. Bailey D, et al. J Am Coll Cardiol. 2010, 55(23), 2580-2589.

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