I-BET151

I-BET151

Product Code: 3432
Availability: In Stock
$3,425.00
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I-BET151 (GSK1210151A) is a novel selective BET inhibitor for BRD2BRD3 and BRD4 with IC50 of 0.5 μM, 0.25 μM, and 0.79 μM, respectively.

Chemical name:

7-(3,5-dimethylisoxazol-4-yl)-8-methoxy-1-((R)-1-(pyridin-2-yl)ethyl)-1H-imidazo[4,5-c]quinolin-2(3H)-one

Biological Activity:
Biological Activity I-BET151 (GSK1210151A) is a novel selective BET inhibitor for BRD2, BRD3 and BRD4 with IC50 of 0.5 μM, 0.25 μM, and 0.79 μM, respectively.
Technical Data:
M.W. 415.44
Formula: <p>C<sub>23</sub>H<sub>21</sub>N<sub>5</sub>O<sub>3</sub></p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 1300031-49-5
References:
References Dawson MA, et al. Nature, 2011, 478(7370), 529-533.

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