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Ki16198

Ki16198

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Product Code: 3410
Availability: In Stock
$461.00
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Ki16198 is the methyl ester of Ki16425, which is a LPAantagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively, shows weaker inhibition for LPA2, no activity at LPA4, LPA5, LPA6.

Chemical Name Propanoic acid, 3-[[[4-[4-[[[1-(2-chlorophenyl)ethoxy]carbonyl]amino]-3-methyl-5-isoxazolyl]phenyl]methyl]thio]-, methyl ester

Inhibitors GPCR & G Protein LPA Receptor Ki16198 355025-13-7
Biological Activity:
Biological Activity Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively, shows weaker inhibition for LPA2, no activity at LPA4, LPA5, LPA6.
Technical Data:
M.W. 488.98
Formula: <p>C<sub>24</sub>H<sub>25</sub>ClN<sub>2</sub>O<sub>5</sub>S</p>
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 355025-13-7
References:
References Komachi M, et al. Cancer Sci, 2012, 103(6), 1099-1104. Shano S, et al. Biochim Biophys Acta, 2008, 1783(5), 748-759. Kimura T, et al. Cardiovasc Res, 2011, 92(1), 149-158.

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